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Bactericidal "isoniazide (INH) #conc-1 rifamacin-2 pyrazinamide-3 cycloserine-$

Bacteriostatic "isoniziade (INH) ! conc-1 ethambuotol-2

Vs Extra & intra cellular organisms -INH 1 Rifampicin-2 ethambutol -3

Extra only streptomycin -1

Intra only Pyrazinamide -1

Enzyme inducer Rifampicin-1 Rifabutin -2

Enzyme inhibitor INH -1

Broad spectrum AB Rifamicin-1 cycloserine-2

Metabolized in liver by acetylation INH-1 %apsone-2

dicated drugs en 1 2 3

oor tolerated &thionamide

E&&ective in typical & atypical 'B 1iprofla+acin 4le*ofla+cin-1 rifabutin-2

'(( 1st line treatment are )i*en !"A##$ e+cept for ,-R&P-./01IN

%tored drugs &thambutol2idney-1 %apsone 2idney 3 s2in3 muscle 4 li*er-2 1lofamazine s2in 4 reticuloendothelial tissues -3 %peci&ic adverse e&&ects -INH peripheral neuritis 3haemolytic anaemia 1 rifampicin harmless oran)e coloration of urine " s5eat 4 contact lens-2 thrombocytopenia3 flu li2e syndrome3 Hyperuricemia 3 6ence-7ones 3induce 1$893 -&thambutol optic neuritis3 hyperuracemia 3 ,treptomycin hyperuracemia 3 .toto+icity 3 Nephroto+icity-$ 1ycloserine peripheral neuropathy 4psychotic reaction-8 (1apreomycin local pain 4 sterile abscess (IV ta2en-: %apsone erythma nodsum-; 1lofamazine &usenic enteritis "red color urine 3s2in discoloration-<

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