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">Priority Number(s):</FONT></TD>

<TD BGCOLOR="#ffffcc"><FONT FACE="Geneva,Arial,Helvetica" SIZE="-1">


<TABLE>
<TR>
<TD><FONT FACE="Geneva,Arial,Helvetica" SIZE="-1">March&nbsp;6,&nbsp;1972</FONT>
</TD>
<TD><FONT FACE="Geneva,Arial,Helvetica" SIZE="-1"><B><A HREF="/details?&pn=GB013
56370A_" MPTYPE="PRIR">GB1972000010439</A></B></FONT></TD>
<TD><FONT FACE="Geneva,Arial,Helvetica" SIZE="-1"><B>
<A HREF="/patlist?&priornumber=GB1972000010439&fullview_selected=CHECKED" MPTYPE
="PRIR">
Family</A></B></FONT>
</TD>
</TR>
</TABLE>
</TD></TR>

<TR
<TD
ca"
<TD

VALIGN="TOP">
WIDTH="129" BGCOLOR="#cccc99" ALIGN="right"><FONT FACE="Geneva,Arial,Helveti
SIZE="-1" COLOR="#996633"><A NAME="ABST"></A>Abstract:</FONT></TD>
WIDTH="402" BGCOLOR="#ffffcc"><FONT FACE="Geneva,Arial,Helvetica" SIZE="-1">

It has been discovered that the unfavorable effects observed in weight reductio
n treatments based on severe dietary restriction (less than 600 Kcals/day) or to
tal fasting (as regards fat, carbohydrates and aminoacids) are avoided by the ad
ministration of aminoacids and carbohydrates in critical but much lower amounts
than has been believed to be necessary. Nitrogen loss with aminoacid intake betw
een about 15 g and 30 g per day is affected by carbohydrate intake. Nitrogen bal
ance is maintained and ketosis and water retention are controlled when the daily
intake includes, in addition to necessary minerals and vitamins, at least 15 g
of
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takes, water retention is absent or minimal. When the carbohydrate intake is inc
reased above about 45 g/day water retention begins to be observable, and with am
ounts above about 75 g/day the water retention may be severe enough to be diagno
sed as clinical edema.
<BR>&#160;&#160;&#160;&#160;In the light of the above discoveries it can be seen
that conventional diets for the treatment of obesity are far from ideal. These
conventional diets are usually prepared from normal food ingredients selected to
be of high protein content, but relatively low in fat and carbohydrate. The nut
rient balance of the preparations may be further adjusted by blending in other f
ood ingredients such as specific proteins isolated from foodstuffs, vitamins and
minerals. Since a diet consisting of protein with some carbohydrate and fat is
not very bulky, non-calorific substances, such as cellulose and methyl cellulose
or similar materials, are sometimes added to provide bulk and hence give a feel
ing of satiety.
<BR>&#160;&#160;&#160;&#160;Usually such conventional diets will give a protein
intake of about 40-60 g/day or more and a carbohydrate intake in excess of 100 g
/day, but so balanced and supplemented with fats as to supply 900-1200 Kcals/day
. Thus these conventional diets supply far larger quantities of protein and carb
ohydrate than the minima now discovered to be necessary. As previously indicated
such conventional formulations suffer from the disadvantages that they cause re
tention of body water due to their high carbohydrate content, and that they are
high in calories, thus slowing down the rate of weight loss. In addition, many o
f them contain the essential and non-essential aminoacids in the wrong proportio
ns.
<BR>&#160;&#160;&#160;&#160;There are other commercially-available food preparat
ions which are not specifically intended for the treatment of obesity, but which
do contain aminoacids present in substantially the proportions required by man-these however all contain more carbohydrate than the above-mentoned optimum.
<BR>&#160;&#160;&#160;&#160;For instance, one such known preparation intended fo
r administration to patients who are to undergo intestinal surgery contains amin
oacids and carbohydrate in a weight ratio of about 1:10. If this preparation wer
e used during severe dietary restriction to treat obesity, in order to satisfy t
he minimum $k 4 ~ VT=]6fL *0Ed 5 /ki,]
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