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I. Muscarinic receptor agonists IV.

Ganglionic stimulants
a. Classification a. Members (3)
i. Choline esters b. Nicotine
1. Acetylcholine
2. Metacholine V. Ganglionic blockers
3. Bethanechol a. Members (3)
4. carbachol b. Effects & uses
ii. Naturally occurring alkaloids
1. Muscarine VI. Adrenergic stimulants
2. Pilocarpine a. Direct acting
3. Arecoline i. Non-selective
b. Therapeutic use (4) ii. Selective
c. Toxicology 1. Alpha 1
2. Alpha 2
II. Muscarinic Receptor Antagonists 3. Beta 1
a. Classification 4. Beta 2
i. Naturally occurring alkaloids b. Inderict acting
1. Atropine i. Releasing agents
2. Scopolamine ii. Uptake inhibitor
ii. Semi-synthetic & synthetic derivatives iii. MAO/COMT inhibitors
1. Omatropine c. Toxicity
2. Tropicamide d. Therapeutic use
3. Methylatropine
4. Ipratropium VII. Adrenergic receptor antagonists
5. Iotropium a. Classification
6. Pirenzepine i. Alpha receptor
7. Tolterodine 1. Non-selective
8. Oxybutynin 2. Alpha 1 selective
b. Pharmacological properties 3. Alpha 2 selective
i. Atropine ii. Beta receptor antagonists
ii. Scopolamine 1. Non-selective
iii. Ipratropium (4) 2. Beta 1
iv. Tiotropium (3) 3. Non-selective
c. Therapeutic use (7) 4. Beta 1
b. Therapeutic use
III. Anti-cholinesterase agents
a. Classification
i. Noncovalent
ii. Reversible carbamate inhibitors
iii. Organophosphorus compounds
b. Pharmacological use
c. Toxicology
d. Therapeutic use

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